Canertinib

Artikelnummer: ENZ-ENZ-CHM196-0005
Artikelname: Canertinib
Artikelnummer: ENZ-ENZ-CHM196-0005
Hersteller Artikelnummer: ENZ-CHM196-0005
Alternativnummer: ENZ-ENZ-CHM196-0005-5
Hersteller: Enzo Life Sciences
Kategorie: Sonstiges
Alternative Synonym: PD-183805, CI-1033, N-[4-[(3-Chloro-4-fluorophenyl)amino]-7-[3-(4-morpholinyl)propoxy]-6-quinazolinyl]-2-propenamide
Canertinib is an orally bio-available EGFR inhibitor with potential anti-neoplastic and radio-sensitizing activities. It has IC50 values of 1.5 nM and 9.0 nM against EGFR and ErbB2 respectively, with no activity against PDGFR, FGFR, InsR, PKC, or CDK1/2/
Molekulargewicht: 485.9
Reinheit: 99% (HPLC)
CAS Nummer: [267243-28-7]
Formel: C24H25ClFN5O3
Target-Kategorie: EGFR, ErbB-2