MLN4924, CAS [[905579-51-3]]

Artikelnummer: FBM-10-1311
Artikelname: MLN4924, CAS [[905579-51-3]]
Artikelnummer: FBM-10-1311
Hersteller Artikelnummer: 10-1311
Alternativnummer: FBM-10-1311-1MG,FBM-10-1311-5MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Alternative Synonym: Pevonedistat
Nedd8 activating enzyme inhibitor
Molekulargewicht: 443.53
Reinheit: 98% by TLC, NMR conforms
Formulierung: White solid
CAS Nummer: [905579-51-3]
Formel: C21H25N5O4S
Anwendungsbeschreibung: Potent and selective NEDD8-activating enzyme (NAE) inhibitor1. It disrupts cullin-RING ligase-mediated protein turnover leading to apoptosis in human tumor cells. Suppresses the growth of human tumor xenografts in mice2. Upregulates PD-L1 expression and