PP242, CAS [[1092351-67-1]]

Artikelnummer: FBM-10-2695
Artikelname: PP242, CAS [[1092351-67-1]]
Artikelnummer: FBM-10-2695
Hersteller Artikelnummer: 10-2695
Alternativnummer: FBM-10-2695-5MG,FBM-10-2695-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Alternative Synonym: Torkinib
Dual mTORC1/mTORC2 inhibitor
Molekulargewicht: 308.35
Reinheit: >98% by HPLC NMR (Conforms)
Formulierung: Off-white to beige solid
CAS Nummer: [1092351-67-1]
Formel: C16H16N6O
Anwendungsbeschreibung: PP242 is an ATP-competitive mTORC1/mTORC2 inhibitor (IC50 = 8 nM) displaying high selectivity over PI 3K family kinases (IC50s =0.102 to 2.2 µM) and modest selectivity over PKC family kinases (IC50s =0.049 to 0.198 µM).1,2 PP 242 (but not rapamycin) indu