EPZ015666, CAS [[1616391-65-1]]

Artikelnummer: FBM-10-4031
Artikelname: EPZ015666, CAS [[1616391-65-1]]
Artikelnummer: FBM-10-4031
Hersteller Artikelnummer: 10-4031
Alternativnummer: FBM-10-4031-5MG,FBM-10-4031-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
PRMT5 inhibitor
Molekulargewicht: 383.44
Reinheit: 98% by HPLC NMR (conforms)
Formulierung: White solid
CAS Nummer: [1616391-65-1]
Formel: C20H25N5O3
Anwendungsbeschreibung: EPZ015666 is a selective and potent (IC50 = 22nM) inhibitor of arginine methyltransferase 5 (PRMT5).1,2 PRMT5 inhibition with EPZ015666 potently suppressed in vivo glioblastoma tumors3 and significantly inhibited the growth of multiple myeloma cell lines