Tazemetostat, CAS [[1403254-99-8]]

Artikelnummer: FBM-10-4032
Artikelname: Tazemetostat, CAS [[1403254-99-8]]
Artikelnummer: FBM-10-4032
Hersteller Artikelnummer: 10-4032
Alternativnummer: FBM-10-4032-5MG,FBM-10-4032-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Alternative Synonym: EPZ-6438
EZH2 inhibitor
Molekulargewicht: 572.75
Reinheit: 98%, NMR (Conforms)
Formulierung: Off-white solid
CAS Nummer: [1403254-99-8]
Formel: C34H44N4O4
Anwendungsbeschreibung: Tazemetostat is a potent (Ki = 2.5nM wild type human PRC2-containing) and selective SAM-competitive inhibitor of the lysine methyltransferase EZH2.1 Tazemetostat displayed strong antiproliferative effects against SMARCB1-deleted malignant rhabdoid tumor