(R)-PFI-2 HCl, CAS [[1627607-87-7]]

Artikelnummer: FBM-10-4033
Artikelname: (R)-PFI-2 HCl, CAS [[1627607-87-7]]
Artikelnummer: FBM-10-4033
Hersteller Artikelnummer: 10-4033
Alternativnummer: FBM-10-4033-5MG,FBM-10-4033-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Methyltransferase SETD7 inhibitor
Molekulargewicht: 535.98
Reinheit: 98% by TLC NMR (Conforms)
Formulierung: White solid
CAS Nummer: [1627607-87-7]
Formel: C23H25F4N3O3S HCl
Anwendungsbeschreibung: Potent (IC50 = 2nM) and selective SAM-dependent inhibitor of the lysine methyltransferase SETD7.1 It alters Hippo pathway signaling in MCF7 cells by altering YAP nuclear localization in a SETD7-dependent manner.