GSK620, CAS [[2088410-46-0]]

Artikelnummer: FBM-10-4047
Artikelname: GSK620, CAS [[2088410-46-0]]
Artikelnummer: FBM-10-4047
Hersteller Artikelnummer: 10-4047
Alternativnummer: FBM-10-4047-5MG,FBM-10-4047-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
BD2 selective BET inhibitor
Molekulargewicht: 325.37
Reinheit: >98% by HPLC NMR (Conforms)
Formulierung: White solid
CAS Nummer: [2088410-46-0]
Formel: C18H19N3O3
Anwendungsbeschreibung: BET inhibitor 220-fold more selective for BD2 over BD1 (pIC50 BD2 = 7.1, BD1 = 4.8).1 It ameliorated collagen-induced arthritis in a rat model and imiquimod-induced psoriasis in a mouse model.2 GSK620 was also able to reduce hepatic fibrosis, steatosis,