ICA-121431, CAS [[313254-51-2]]

Artikelnummer: FBM-10-4085
Artikelname: ICA-121431, CAS [[313254-51-2]]
Artikelnummer: FBM-10-4085
Hersteller Artikelnummer: 10-4085
Alternativnummer: FBM-10-4085-5MG,FBM-10-4085-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Nav1.1/1.3 inhibitor (selective)
Molekulargewicht: 449.54
Reinheit: 98% by TLC , NMR (Conforms)
Formulierung: Off-white to beige solid
CAS Nummer: [313254-51-2]
Formel: C23H19N3O3S2
Anwendungsbeschreibung: Selective Nav1.1/1.3 inhibitor (hIC50s = 23 and 13 nM respectively, also selective for dog, monkey, and mouse, but not rat).1 It exclusively shifts voltage dependence to more negative voltages and accelerates entry into slow activation.2