MF-438, CAS [[921605-87-0]]

Artikelnummer: FBM-10-4558
Artikelname: MF-438, CAS [[921605-87-0]]
Artikelnummer: FBM-10-4558
Hersteller Artikelnummer: 10-4558
Alternativnummer: FBM-10-4558-5MG,FBM-10-4558-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
SCD1 inhibitor
Molekulargewicht: 421.44
Reinheit: 98% by HPLC, NMR (Confirms)
Formulierung: Off-white solid
CAS Nummer: [921605-87-0]
Formel: C19H18F3N5OS
Anwendungsbeschreibung: MF-438 is a potent inhibitor of stearoyl-CoA desaturase 1 (SCD1) - IC50 = 2.3 nM.1 MF-438 was potent in an in vivo mouse liver PD assay (ED50 between 1 and mg/kg).1 Cancer initiating cells (CSC-like) were shown to much more sensitive to MF-438 inhibition