Trametinib, CAS [[871700-17-3]]

Artikelnummer: FBM-10-4759
Artikelname: Trametinib, CAS [[871700-17-3]]
Artikelnummer: FBM-10-4759
Hersteller Artikelnummer: 10-4759
Alternativnummer: FBM-10-4759-10MG,FBM-10-4759-50MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Alternative Synonym: GSK1120212, JTP-74057
MEK inhibitor
Molekulargewicht: 615.39
Reinheit: 98% by TLC/HPLC NMR (Conforms)
Formulierung: White solid
CAS Nummer: [871700-17-3]
Formel: C26H23FIN5O4
Anwendungsbeschreibung: Trametinib is a highly potent (IC50 uMEK1 = 0.7 nM, pp-MEK1 = 14.9 nM)1 and selective MEK inhibitor displaying selective inhibition of proliferation in various BRAF mutant cancer cell lines (IC50 ACHN = 9.8 nM, IC50 HT-29 = 0.57 nM)2. It is approved for