Binimetinib, CAS [[606143-89-9]]

Artikelnummer: FBM-10-4789
Artikelname: Binimetinib, CAS [[606143-89-9]]
Artikelnummer: FBM-10-4789
Hersteller Artikelnummer: 10-4789
Alternativnummer: FBM-10-4789-5MG,FBM-10-4789-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Alternative Synonym: ARRY-162, MEK162
MEK1/2 inhibitor
Molekulargewicht: 441.23
Reinheit: 99% by HPLC NMR (Conforms)
Formulierung: White solid
CAS Nummer: [606143-89-9]
Formel: C17H15BrF2N4O3
Anwendungsbeschreibung: Binimetinib (606143-89-9) is a potent (IC50 = 12 nM) and selective allosteric inhibitor of MEK1/2.1,2 Recently approved by the FDA for treatment of melanoma in combination with Encorafenib. Binimetinib has had limited success as monotherapy but has shown