Pexidartinib, CAS [[1029044-16-3]]

Artikelnummer: FBM-10-4829
Artikelname: Pexidartinib, CAS [[1029044-16-3]]
Artikelnummer: FBM-10-4829
Hersteller Artikelnummer: 10-4829
Alternativnummer: FBM-10-4829-5MG,FBM-10-4829-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Alternative Synonym: PLX3397
CSF1R inhibitor
Molekulargewicht: 417.81
Reinheit: 98% by HPLC NMR (Conforms)
Formulierung: White solid
CAS Nummer: [1029044-16-3]
Formel: C20H15ClF3N5
Anwendungsbeschreibung: Pexidartinib (1029044-16-3) is a potent and selective dual inhibitor of CSF1R (IC50 = 20nM) and c-KIT (IC50 = 10nM).1 Inhibition of CSF1R with Pexidartinib resulted in a reprogrammed immune microenvironment that fosters antitumor immunity in a CD8+ T-cel