GSK2656157, CAS [[1337532-29-2]]

Artikelnummer: FBM-10-4855
Artikelname: GSK2656157, CAS [[1337532-29-2]]
Artikelnummer: FBM-10-4855
Hersteller Artikelnummer: 10-4855
Alternativnummer: FBM-10-4855-5MG,FBM-10-4855-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Potent and selective PERK inhibitor
Molekulargewicht: 416.45
Reinheit: 98% by HPLC NMR (Conforms)
Formulierung: White solid
CAS Nummer: [1337532-29-2]
Formel: C23H21FN6O
Anwendungsbeschreibung: Potent (IC50 = 0.9 nM) and selective (over 300 kinases) inhibitor of protein kinase RNA-like endoplasmic reticulum kinase (PERK).1,2 Inhibited growth of multiple human tumor xenografts in mice. GSK2656157 has also been found to potently inhibit RIPK1 (IC