SX-682, CAS [[1648843-04-2]]

Artikelnummer: FBM-10-4925
Artikelname: SX-682, CAS [[1648843-04-2]]
Artikelnummer: FBM-10-4925
Hersteller Artikelnummer: 10-4925
Alternativnummer: FBM-10-4925-5MG,FBM-10-4925-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
CXCR1/2 inhibitor
Molekulargewicht: 467.20
Reinheit: 98% by HPLC NMR (Conforms)
Formulierung: Off-white solid
CAS Nummer: [1648843-04-2]
Formel: C19H14BF4N3O4S
Anwendungsbeschreibung: SX-682 is a novel CXCR1/2 inhibitor (IC50s: CXCR1 = 42 nM, CXCR2 = 20 nM)1. It displayed robust synergistic activity with immune checkpoint blockade against castration resistant prostate cancer.2 It significantly reduced tumor burden in a Ptenfl/fl/Lkb1f