GKT-137831, CAS [[1218942-37-0]]

Artikelnummer: FBM-10-5044
Artikelname: GKT-137831, CAS [[1218942-37-0]]
Artikelnummer: FBM-10-5044
Hersteller Artikelnummer: 10-5044
Alternativnummer: FBM-10-5044-5MG,FBM-10-5044-25MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Alternative Synonym: Setanaxib, GKT-831
NADPH oxidase NOX1/4 inhibitor
Molekulargewicht: 394.85
Reinheit: 98% by TLC NMR (Conforms)
Formulierung: Pale-yellow solid
CAS Nummer: [1218942-37-0]
Formel: C21H19ClN4O2
Anwendungsbeschreibung: NADPH oxidase, NOX1/4 inhibitor (Ki = 100-150 nM).1 Inhibits erastin-stimulated ROS production.2 Potentiates immunotherapy by overcoming cancer-associated fibroblast- mediated CD8+ T-cell exclusion.3 Reduces ROS production in LPS-stimulated platelets in