Samuraciclib (hydrochloride dihydrate)

Artikelnummer: MCE-HY-103712B
Artikelname: Samuraciclib (hydrochloride dihydrate)
Artikelnummer: MCE-HY-103712B
Hersteller Artikelnummer: HY-103712B
Alternativnummer: MCE-HY-103712B-5MG,MCE-HY-103712B-25MG,MCE-HY-103712B-100MG,MCE-HY-103712B-10MG,MCE-HY-103712B-50MG,MCE-HY-103712B-10MMX1ML
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: CT7001 (hydrochloride dihydrate), ICEC0942 (hydrochloride dihydrate)
Samuraciclib (CT7001) hydrochloride hydrate is a potent, selective, ATP-competitive and orally active CDK7 inhibitor, with an IC50 of 41 nM. Samuraciclib hydrochloride hydrate displays 45-, 15-, 230- and 30-fold selectivity over CDK1, CDK2 (IC50 of 578 n
Molekulargewicht: 521.70
Reinheit: 99.08
Formel: C22H30N6O.(2.5HCl).(2H2O)
Target-Kategorie: Apoptosis,CDK
Anwendungsbeschreibung: Reference compound