Samuraciclib (hydrochloride hydrate)

Artikelnummer: MCE-HY-103712C
Artikelname: Samuraciclib (hydrochloride hydrate)
Artikelnummer: MCE-HY-103712C
Hersteller Artikelnummer: HY-103712C
Alternativnummer: MCE-HY-103712C-25MG,MCE-HY-103712C-5MG,MCE-HY-103712C-100MG,MCE-HY-103712C-10MMX1ML,MCE-HY-103712C-50MG,MCE-HY-103712C-10MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: CT7001 (hydrochloride hydrate), ICEC0942 (hydrochloride hydrate)
Samuraciclib (CT7001) hydrochloride hydrate is a potent, selective, ATP-competitive and orally active CDK7 inhibitor, with an IC50 of 41 nM. Samuraciclib hydrochloride hydrate displays 45-, 15-, 230- and 30-fold selectivity over CDK1, CDK2 (IC50 of 578 n
Molekulargewicht: 552.33
Reinheit: 99.88
Formel: C22H30N6O.(2.5HCl).(3.7H2O)
Target-Kategorie: Apoptosis,CDK
Anwendungsbeschreibung: Reference compound