Glumetinib (SCC244) is a highly selective, orally bioavailable, ATP-competitive c-Met inhibitor with an IC50 of 0.42 nM. Glumetinib has greater than 2400-fold selectivity for c-Met over those 312 kinases evaluated, including the c-Met family member RON a
Molekulargewicht:
459.48
Reinheit:
99.92
CAS Nummer:
[1642581-63-2]
Formel:
C21H17N9O2S
Target-Kategorie:
c-Met/HGFR
Anwendungsbeschreibung:
Reference compound
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