Multi-kinase-IN-4 (compound 5d) is multi-targeted kinase inhibitor, including VEGFR2, EGFR, HER2, and CDK2, with IC50 values of 0.33, 0.22, 0.18 and 2.09 µM, respectively. Multi-kinase-IN-4 shows broad-spectrum anti-cancer activities against HepG2, MCF-7
Molekulargewicht:
402.91
Formel:
C21H20ClFN2OS
Target-Kategorie:
Apoptosis,CDK,EGFR,Necroptosis,VEGFR
Anwendungsbeschreibung:
Reference compound
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