PBRM1-BD2-IN-8, CAS [[2819989-75-6]]
Artikelnummer:
MCE-HY-151538
Artikelname: |
PBRM1-BD2-IN-8, CAS [[2819989-75-6]] |
Artikelnummer: |
MCE-HY-151538 |
Hersteller Artikelnummer: |
HY-151538 |
Alternativnummer: |
MCE-HY-151538-1MG |
Hersteller: |
MedchemExpress |
Kategorie: |
Biochemikalien |
PBRM1-BD2-IN-8 (compound 34) is a potent PBRM1 Bromodomain inhibitor (PBRM1-BD2 Kd=4.4 µM, PBRM1-BD2 IC50=0.16 µM, PBRM1-BD5 Kd=25 µM). PBRM1-BD2-IN-8 shows anti-cancer activity[1]. |
Molekulargewicht: |
317.18 |
Reinheit: |
99.48 |
CAS Nummer: |
[2819989-75-6] |
Formel: |
C15H13BrN2O |
Target-Kategorie: |
Epigenetic Reader Domain |
Anwendungsbeschreibung: |
Reference compound |