TRK-IN-24 (compound 10g) is a Trk Receptor inhibitor that inhibits TRKA, TRKC, TRKAG595R, TRKAG667C and TRKAF589L IC50s are 5.21, 4.51, 6.77, 1.42 and 6.13 nM respectively. TRK-IN-24 has antitumor efficacy in BaF3-CD74-NTRK1G595R and BaF3-CD74-NTRK1G667C
Molekulargewicht:
659.82
CAS Nummer:
[2937544-01-7]
Formel:
C39H45N7O3
Target-Kategorie:
Trk Receptor
Anwendungsbeschreibung:
Reference compound
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