GSK-J4 (hydrochloride), CAS [[1797983-09-5]]

Artikelnummer: MCE-HY-15648F
Artikelname: GSK-J4 (hydrochloride), CAS [[1797983-09-5]]
Artikelnummer: MCE-HY-15648F
Hersteller Artikelnummer: HY-15648F
Alternativnummer: MCE-HY-15648F-50MG,MCE-HY-15648F-5MG,MCE-HY-15648F-10MMX1ML,MCE-HY-15648F-10MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
GSK-J4 hydrochloride is a potent dual inhibitor of H3K27me3/me2-demethylases JMJD3/KDM6B and UTX/KDM6A with IC50s of 8.6 and 6.6 µM, respectively. GSK-J4 hydrochloride inhibits LPS-induced TNF-alpha production in human primary macrophages with an IC50 of 9 µ
Molekulargewicht: 453.96
Reinheit: 98.83
CAS Nummer: [1797983-09-5]
Formel: C24H28ClN5O2
Target-Kategorie: Histone Demethylase
Anwendungsbeschreibung: Reference compound