GDC-0152
Artikelnummer:
SEL-S7010
- Bilder (0)
Artikelname: | GDC-0152 |
Artikelnummer: | SEL-S7010 |
Hersteller Artikelnummer: | S7010 |
Alternativnummer: | SEL-S7010-10MG,SEL-S7010-10MM/1ML,SEL-S7010-100MG |
Hersteller: | Selleck |
Kategorie: | Biochemikalien |
GDC-0152 is a potent antagonist of XIAP-BIR3, ML-IAP-BIR3, cIAP1-BIR3 and cIAP2-BIR3 with Ki of 28 nM, 14 nM, 17 nM and 43 nM in cell-free assays, respectively, less affinity shown to cIAP1-BIR2 and cIAP2-BIR2. Phase 1. |
CAS Nummer: | [873652-48-3] |