Pelabresib (CPI-0610)
Artikelnummer:
SEL-S7853
- Bilder (0)
Artikelname: | Pelabresib (CPI-0610) |
Artikelnummer: | SEL-S7853 |
Hersteller Artikelnummer: | S7853 |
Alternativnummer: | SEL-S7853-10MM/1ML,SEL-S7853-100MG,SEL-S7853-25MG,SEL-S7853-5MG |
Hersteller: | Selleck |
Kategorie: | Biochemikalien |
Pelabresib (CPI-0610) is a potent and selective benzoisoxazoloazepine BET bromodomain inhibitor with an IC50 of 39 nM for BRD4-BD1 in TR-FRET assay and currently undergoing human clinical trials for hematological malignancies. CPI-0610 inhibits the expre |