Pelabresib (CPI-0610)

Artikelnummer: SEL-S7853
Artikelname: Pelabresib (CPI-0610)
Artikelnummer: SEL-S7853
Hersteller Artikelnummer: S7853
Alternativnummer: SEL-S7853-10MM/1ML,SEL-S7853-100MG,SEL-S7853-25MG,SEL-S7853-5MG
Hersteller: Selleck
Kategorie: Biochemikalien
Pelabresib (CPI-0610) is a potent and selective benzoisoxazoloazepine BET bromodomain inhibitor with an IC50 of 39 nM for BRD4-BD1 in TR-FRET assay and currently undergoing human clinical trials for hematological malignancies. CPI-0610 inhibits the expre