Tropifexor (LJN452)

Artikelnummer: SEL-S8733
Artikelname: Tropifexor (LJN452)
Artikelnummer: SEL-S8733
Hersteller Artikelnummer: S8733
Alternativnummer: SEL-S8733-10MG,SEL-S8733-2MG
Hersteller: Selleck
Kategorie: Biochemikalien
Tropifexor (LJN452) is a novel and highly potent agonist of FXR with EC50 of 0.2 nM in HTRF assay. It shows no significant off-target activity against a broad panel of enzyme, ion channel, nuclear receptor, and GPCR (>10000-fold selectivity for FXR).
CAS Nummer: [1383816-29-2]