YKL-5-124
Artikelnummer:
SEL-S8863
- Bilder (0)
Artikelname: | YKL-5-124 |
Artikelnummer: | SEL-S8863 |
Hersteller Artikelnummer: | S8863 |
Alternativnummer: | SEL-S8863-10MM/1ML,SEL-S8863-25MG,SEL-S8863-5MG |
Hersteller: | Selleck |
Kategorie: | Biochemikalien |
YKL-5-124 is a potent, selective and covalent CDK7 inhibitor with an IC50 of 9.7 nM, 1300 nM and 3020 nM for inhibiting CDK7/Mat1/CycH, CDK2 and CDK9 respectively. It displays biochemical and cellular selectivity for CDK7 over CDK12/13. |
CAS Nummer: | [1957203-01-8] |