LT052, CAS [[2543545-44-2]]

Artikelnummer: TGM-T11887
Artikelname: LT052, CAS [[2543545-44-2]]
Artikelnummer: TGM-T11887
Hersteller Artikelnummer: T11887
Alternativnummer: TGM-T11887-25MG,TGM-T11887-50MG
Hersteller: TargetMol
Kategorie: Biochemikalien
LT052, a highly active and selective BET BD1 inhibitor with an IC50 of 87.7 nM, demonstrates nanomolar BRD4 BD1 potency and significant selectivity, being 138-fold more selective for BRD4 BD1 over BRD4 BD2 (IC50 =12.130 µM). Its anti-inflammatory propert
Molekulargewicht: 449.48
CAS Nummer: [2543545-44-2]
Formel: C22H19N5O4S
Target-Kategorie: Epigenetic Reader Domain