TC-MCH 7c is an oral, selectable and blood-brain barrier penetrating MCH1R antagonist with IC50 performance of 5.6 nM against hMCH1R, and TC-MCH 7c is a phenylpyridone derivative with MCH1R Ki of 3.4 nM against human. In mice, MCH1R Ki was 3.0 nM.
Molekulargewicht:
408.47
CAS Nummer:
[864756-35-4]
Formel:
C24H25FN2O3
Target-Kategorie:
Melanin-concentrating Hormone Receptor (MCHR)
T13101
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