Alpelisib, CAS [[1217486-61-7]]
Artikelnummer:
TGM-T1921
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Artikelname: | Alpelisib, CAS [[1217486-61-7]] |
Artikelnummer: | TGM-T1921 |
Hersteller Artikelnummer: | T1921 |
Alternativnummer: | TGM-T1921-1G,TGM-T1921-1ML,TGM-T1921-5MG,TGM-T1921-10MG,TGM-T1921-25MG,TGM-T1921-50MG,TGM-T1921-100MG,TGM-T1921-200MG,TGM-T1921-500MG |
Hersteller: | TargetMol |
Kategorie: | Biochemikalien |
Alternative Synonym: | BYL-719 |
Alpelisib (BYL-719) is a PI3Kalpha inhibitor (IC50=5 nM) with selective, potent, and oral activity, inhibiting PI3Kbeta/gamma/delta with low activity (IC50=250/290/1200 nM). Alpelisib demonstrates antitumor activity and specifically targets PIK3CA mutant tumors. |
Molekulargewicht: | 441.47 |
CAS Nummer: | [1217486-61-7] |
Formel: | C19H22F3N5O2S |
Target-Kategorie: | PI3K |