PF 05089771 tosylate, CAS [[1430806-04-4]]

Artikelnummer: TGM-T7502
Artikelname: PF 05089771 tosylate, CAS [[1430806-04-4]]
Artikelnummer: TGM-T7502
Hersteller Artikelnummer: T7502
Alternativnummer: TGM-T7502-1MG,TGM-T7502-5MG,TGM-T7502-10MG,TGM-T7502-25MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: (S)-(4-((5-Fluoro-4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)pyrimidin-2-yl)amino)phenyl)(3-(methylamino)pyrrolidin-1-yl)methanone
PF-05089771 is a voltage-gated sodium channel 1.7 (Nav1.7) blocker (IC50: 11, 16, 33, and 20 nM for 5N11S, 5A11L, 5A11S, and 5A11L Nav1.7 splice variants, respectively). It is selective for Nav1.7 over Nav1.1-1.6 and 1.8 channels (IC50: 0.11-25 µM), L-ty
Molekulargewicht: 672.56
CAS Nummer: [1430806-04-4]
Formel: C18H12Cl2FN5O3S2.C7H8O3S