YXG-158 (Compound 23-h), an orally active androgen receptor (AR) degrader and cytochrome P450 17A1 (CYP17A1) inhibitor, exhibits AR degradation with a DC50 of 1.28 µM and CYP17A1 inhibition with an IC50 of 100 nM. It is under investigation for potential
Molekulargewicht:
473.62
CAS Nummer:
[2952994-34-0]
Formel:
C30H36FN3O
Target-Kategorie:
Androgen Receptor
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