GSK2193874 is a first-in-class orally bioavailable potent antagonist of TRPV4 channels, blocking the influx of calcium induced by the TRPV4 agonist with IC50 values of 2, 5, and 40 nM. GSK2193874 is the first-in-class orally bioavailable TRPV4 inhibitor
Molecular Weight:
691.62
Purity:
>99%
CAS Number:
[1336960-13-4]
Formula:
C37H38BrF3N4O
Target:
TRP Channel
* VAT and and shipping costs not included. Errors and price changes excepted