Gambogenic acid is the active ingredient in Huangteng and has anti-cancer activity. Gambogenic acid is an effective EZH2 inhibitor, which specifically covalently binds to Cys668 in the EZH2-SET domain to induce EZH2 ubiquitination.
Molecular Weight:
630.78
Purity:
>99%
CAS Number:
[173932-75-7]
Formula:
C38H46O8
Target:
Histone Methyltransferase
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