Cpi-169 (CPI 169 R-Enantiomer) is a novel and effective EZH2 inhibitor, capable of inhibiting the activity of EZH2 WT, EZH2 Y641N and EZH1 with IC50 value of 0.24 nM, respectively. 0.51 nM and 6.1 nM.
Molecular Weight:
528.66
Purity:
>98%
CAS Number:
[1802175-07-0]
Formula:
C27H36N4O5S
Target:
Histone Methyltransferase
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