Gartisertib (VX-803) is an ATP-competitive, orally active, selective ATR inhibitor with Ki<150 pM. Gartisertib inhibits atR-driven phosphorylation of checkpoint kinase-1 (Chk1) with an IC50 value of 8 nM. It has antitumor activity.
Molecular Weight:
541.55
Purity:
>99%
CAS Number:
[1613191-99-3]
Formula:
C25H29F2N9O3
Target:
ATM/ATR
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