LE135 is an effective RAR antagonist, which can selectively bind RARalpha (Ki is 1.4 µM) and RARbeta (Ki is 220 nM), and has a higher affinity for RARbeta. The LE135 is highly selective for RARgamma, RXRalpha, RXRbeta and RXRgamma. LE135 is also a vitamin A acid receptor antagon
Molecular Weight:
438.56
Purity:
>99%
CAS Number:
[155877-83-1]
Formula:
C29H30N2O2
Target:
RAR/RXR
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