Tenalisib (RP6530) is a potent and selective dual PI3Kdelta/gamma inhibitor with IC50 values of 24.5 nM and 33.2 nM for PI3Kdelta and PI3Kgamma, respectively. Its selectivity over alpha and beta isoforms are more than 300-fold and 100-fold, respectively.
Molecular Weight:
415.42
Purity:
>98.0%
CAS Number:
[1639417-53-0]
Formula:
C23H18FN5O2
Target:
PI3K
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