PLX51107 is a potent and selective BET inhibitor, with Kds of 1.6, 2.1, 1.7, and 5 nM for BD1 and 5.9, 6.2, 6.1, and 120 nM for BD2 of BRD2, BRD3, BRD4, and BRDT, respectively.
Molecular Weight:
438.48
Purity:
>99%
CAS Number:
[1627929-55-8]
Formula:
C26H22N4O3
Target:
Epigenetic Reader Domain
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