Selpercatinib (LOXO-292) is a first-in-class, highly selective and potent small molecule RET inhibitor with good blood-brain barrier (BBB) penetration. and RET (G810R) with IC50 values of 14.0 nM, 24.1 nM and 530.7 nM, respectively.
Molecular Weight:
525.6
Purity:
99.98%
CAS Number:
[2152628-33-4]
Formula:
C29H31N7O3
Target:
RET
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