Canertinib is an orally bio-available EGFR inhibitor with potential anti-neoplastic and radio-sensitizing activities. It has IC50 values of 1.5 nM and 9.0 nM against EGFR and ErbB2 respectively, with no activity against PDGFR, FGFR, InsR, PKC, or CDK1/2/
Molecular Weight:
485.9
Purity:
99% (HPLC)
CAS Number:
[267243-28-7]
Formula:
C24H25ClFN5O3
Target:
EGFR, ErbB-2
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