CB-839, CAS [[1439399-58-2]]

Product Overview

• Article Name: CB-839, CAS [[1439399-58-2]]
• Biozol Catalog Number: FBM-10-4556
• Supplier Catalog Number: 10-4556
• Alternative Catalog Number: FBM-10-4556-5MG,FBM-10-4556-25MG
• Manufacturer: Focus Biomolecules
• Category: Biochemikalien
• Alternative Names: Telaglenastat

Product Description

Glutaminase inhibitor

Product Properties

• Molecular Weight: 571.57
• Purity: >97% by HPLC: Agilent Poroshell 120 C18, 80/20 MeOH/water, 0.8 mL/min, 245 and 270 nm. NMR (Conforms)
• Form: Pale yellow solid
• CAS Number: [1439399-58-2]
• Formula: C26H24F3N7O3S

Application Notes

• Application Notes: CB-839 is a potent (IC50 = 24 nM), selective and orally bioavailable inhibitor of glutaminase (KGA and GAC).1 CB-839 displayed an antiproliferative effect in the triple-negative breast cancer cell line, HCC-1806, but no activity in the estrogen receptor-