1G244, CAS [[847928-32-9]]

Product Overview

• Article Name: 1G244, CAS [[847928-32-9]]
• Biozol Catalog Number: FBM-10-4584
• Supplier Catalog Number: 10-4584
• Alternative Catalog Number: FBM-10-4584-5MG,FBM-10-4584-25MG
• Manufacturer: Focus Biomolecules
• Category: Biochemikalien
• Alternative Names: PTX-1210

Product Description

DPP8/9 inhibitor

Product Properties

• Molecular Weight: 504.57
• Purity: >98% by HPLC, NMR (Conforms)
• Form: Off-white solid
• CAS Number: [847928-32-9]
• Formula: C29H30F2N4O2

Application Notes

• Application Notes: Potent and selective inhibitor of the prolyl dipeptidases DPP8 (IC50 = 14 nM) and DPP9 (IC50 = 53 nM).1,2 It does not inhibit DPP2, DPP4 or fibroblast activation protein (FAP) at 100 µM.1,2 1G244 is a slow binding competitive inhibitor of DPP8 but a comp