GSK2656157, CAS [[1337532-29-2]]

Product Overview

• Article Name: GSK2656157, CAS [[1337532-29-2]]
• Biozol Catalog Number: FBM-10-4855
• Supplier Catalog Number: 10-4855
• Alternative Catalog Number: FBM-10-4855-5MG,FBM-10-4855-25MG
• Manufacturer: Focus Biomolecules
• Category: Biochemikalien

Product Description

Potent and selective PERK inhibitor

Product Properties

• Molecular Weight: 416.45
• Purity: 98% by HPLC NMR (Conforms)
• Form: White solid
• CAS Number: [1337532-29-2]
• Formula: C23H21FN6O

Application Notes

• Application Notes: Potent (IC50 = 0.9 nM) and selective (over 300 kinases) inhibitor of protein kinase RNA-like endoplasmic reticulum kinase (PERK).1,2 Inhibited growth of multiple human tumor xenografts in mice. GSK2656157 has also been found to potently inhibit RIPK1 (IC