SX-682, CAS [[1648843-04-2]]

Catalog Number: FBM-10-4925
Article Name: SX-682, CAS [[1648843-04-2]]
Biozol Catalog Number: FBM-10-4925
Supplier Catalog Number: 10-4925
Alternative Catalog Number: FBM-10-4925-5MG,FBM-10-4925-25MG
Manufacturer: Focus Biomolecules
Category: Biochemikalien
CXCR1/2 inhibitor
Molecular Weight: 467.20
Purity: 98% by HPLC NMR (Conforms)
Form: Off-white solid
CAS Number: [1648843-04-2]
Formula: C19H14BF4N3O4S
Application Notes: SX-682 is a novel CXCR1/2 inhibitor (IC50s: CXCR1 = 42 nM, CXCR2 = 20 nM)1. It displayed robust synergistic activity with immune checkpoint blockade against castration resistant prostate cancer.2 It significantly reduced tumor burden in a Ptenfl/fl/Lkb1f