Varenicline (CP 526555) is an orally active partial agonist of alpha4beta2 nicotinic acetylcholine receptor (alpha4beta2 nAChR, IC50 = 250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of alpha6beta2 nAChR and a full agoni
Molecular Weight:
211.26
Purity:
99.98
CAS Number:
[249296-44-4]
Formula:
C13H13N3
Target:
nAChR
Application Notes:
Reference compound
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