Varenicline (CP 526555-18) is an orally active partial agonist of alpha4beta2 nicotinic acetylcholine receptor (alpha4beta2 nAChR, IC50 = 250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of alpha6beta2 nAChR and a full ag
Molecular Weight:
284.18
Purity:
99.21
CAS Number:
[866823-63-4]
Formula:
C13H15Cl2N3
Target:
nAChR
Application Notes:
Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted