Ruboxistaurin (LY333531) is an orally active, selective PKC beta inhibitor (Ki=2 nM). Ruboxistaurin exhibits ATP dependent competitive inhibition of PKC beta I with an IC50 of 4.7 nM. Ruboxistaurin inhibits PKC beta II with an IC50 of 5.9 nM[1][2].
Molecular Weight:
468.55
Purity:
99.90
CAS Number:
[169939-94-0]
Formula:
C28H28N4O3
Target:
PKC
Application Notes:
Reference compound
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