Samuraciclib (hydrochloride hydrate)

Catalog Number: MCE-HY-103712C
Article Name: Samuraciclib (hydrochloride hydrate)
Biozol Catalog Number: MCE-HY-103712C
Supplier Catalog Number: HY-103712C
Alternative Catalog Number: MCE-HY-103712C-25MG,MCE-HY-103712C-5MG,MCE-HY-103712C-100MG,MCE-HY-103712C-10MMX1ML,MCE-HY-103712C-50MG,MCE-HY-103712C-10MG
Manufacturer: MedchemExpress
Category: Biochemikalien
Alternative Names: CT7001 (hydrochloride hydrate), ICEC0942 (hydrochloride hydrate)
Samuraciclib (CT7001) hydrochloride hydrate is a potent, selective, ATP-competitive and orally active CDK7 inhibitor, with an IC50 of 41 nM. Samuraciclib hydrochloride hydrate displays 45-, 15-, 230- and 30-fold selectivity over CDK1, CDK2 (IC50 of 578 n
Molecular Weight: 552.33
Purity: 99.88
Formula: C22H30N6O.(2.5HCl).(3.7H2O)
Target: Apoptosis,CDK
Application Notes: Reference compound