Talmapimod (SCIO-469) is an orally active, selective, and ATP-competitive p38alpha inhibitor with an IC50 of 9 nM. Talmapimod shows about 10-fold selectivity over p38beta, and at least 2000-fold selectivity over a panel of 20 other kinases, including other MAPK
Molecular Weight:
513.00
Purity:
98.97
CAS Number:
[309913-83-5]
Formula:
C27H30ClFN4O3
Target:
p38 MAPK
Application Notes:
Reference compound
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