TG101209 is a selective JAK2 inhibitor with IC50 of 6 nM, less potent to Flt3 and RET with IC50 of 25 nM and 17 nM, appr 30-fold selective for JAK2 than JAK3, and sensitive to JAK2V617F and MPLW515L/K mutations.
Molecular Weight:
509.67
Purity:
99.22
CAS Number:
[936091-14-4]
Formula:
C26H35N7O2S
Target:
Apoptosis,Autophagy,FLT3,JAK,RET
Application Notes:
Reference compound
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